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Richard J. Prankerd
Senior Lecturer in Pharmaceutics
BPharm, MPharm, PhD, Univ. Otago
Phone: +61 3 9903 9003
Fax: +61 3 9903 9583
Email: Richard.Prankerd@pharm.monash.edu.au
General Research Interests
- Physical and pharmaceutical chemistry
- Solution equilibria and kinetics
- Thermal analysis and spectroscopy
- Analytical methods development
- Formulation science
Current Research Areas
- Applications of solution microcalorimetry in pharmaceutical and formulation science. (This work currently involves on-campus collaborations with Profs. W. Charman and C. Pouton, Assoc Profs. S. Charman and C. Porter, and Drs. M. Scanlon and D. Warren; off-campus collaborations with Dr. John Forsyth, Monash Clayton, and Dr Ross Kennedy, Charles Sturt Uni)
- Characterisation and pharmaceutical evaluation of a novel natural product gum. (Dr U.U. Ben-Nwauzor)
- Development of novel gene transfection agents (collaboration with Prof. C. Pouton and Dr. J. Jazayeri)
Honours projects for 2008
Significant Publications
- Prankerd, R.J. Critical compilation of PKA values for pharmaceutical substances. (2007) Profiles of drug substances, excipients, and related methodology 33.
- Horner, J., d'Auvergne, E.J., Coles, M., Velkov, T., Chin, Yanni., Charman, W.N., Prankerd, R., Gooley, P.R., Scanlon, M.J. Probing the flexibility of the DsbA oxidoreductase from vibrio cholerae -a 15N – 1H heteronuclear NMR relaxation analysis of oxidized and reduced forms of DsbA. (2007) Journal of Molecular Biology 371, 703-716.
- Creek, J.D., Charman, W.N., Chiu, F.C.K., Prankerd, R.J., McCullough, K.J., Dong, Y., Vennerstrom, J.L., Charman, S.A. Iron-mediated degredation kinetics of substituted dispiro-1,2,4-trioxolane antimalarials. (2007) Journal of Pharmaceutical Sciences 96(11) 2945-2956.
- Perry, C., Charman, S.A., Prankerd, R.J., Chiu, F., Dong, Y., Vennerstrom, J. and Charman, W.N. Chemical kinetics and aqueous degradation pathways of a new class of synthetic ozonide antimalarials. (2006) Journal of Pharmaceutical Sciences 95(4): 373-747.
- Perry, C., Charman, S.A., Prankerd, R.J., Chiu, F., Scanlon, M., Chalmers, D. and Charman. W.N. The binding interaction of synthetic ozonide antimalarials with natural and modified ß-cyclodextrins. (2006) Journal of Chromatography B 830: 314-321.
- Charman, S.A., Perry, C., Chiu, F., McIntosh, K., Prankerd, R.J., Charman, W.N. Alteration of the intravenous pharmacokinetics of a synthetic ozonide antimalarial in the presence of a modified cyclodextrin. (2006) Journal of Pharmaceutical Sciences 95(2): 256-267.
- Velkov, T., Chuang, S., Prankerd, R., Sakellaris, H., Porter, C.J.H. and Scanlon, M. An improved method for the purification of rat liver-type fatty acid binding protein from Escherichia coli. Protein Expression & Purification 44 23-31 (2005)
- Creek, D.J., Chiu, F., Prankerd, P., Charman, S.A. and Charman, W.N. Kinetics of iron-mediated artemisinin degradation: effect of solvent composition and iron salt. J. Pharm. Sci., 94: 1820-1829 (2005).
- Ben-Nwauzor, U.U. and Prankerd R.J., Isolation and studies on the chemical composition and structural characteristics of novel polysaccharide mucilage from the calyx of Bombax costatum. Carbohydrate Research, (2004).
- Davie, A.S., Campbell, M., Prankerd, R.J. and Charman, W.N. Stability of berenil in acidic aqueous solutions. J Pharm. Pharmacol. Vol. 56, No. 10 pp.1327-1332, (2004)
- Taillardat-Bertschinger, A., Perry,C.S., Galland, A., Prankerd, R.J. and Charman, W.N. Partitioning of halofantrine hydrochloride between water, micellar solutions and soybean oil: Effects on its apparent ionization constant. J.Pharm.Sci. 92 (11) 2217-28, (2003)
- Khoo, S.M., Prankerd, R. J., Edwards,G. A., Porter, C.J.H. and Charman, W. N. A physicochemical basis for the significant intestinal lymphatic transport of a poorly lipid soluble antimalarial, halofantrine hydrochloride, after post-prandial administration. J.Pharm.Sci. 91, 647-659, (2003)
- Shackleford, D., Prankerd, R.J., Scanlon, M.J. and Charman, W.N. Self-micellization of Gemfibrozil 1-O-β Acyl Glucuronide in aqueous solution. Pharm. Res. 20(3) 465-470 2003.
- Prankerd, R.J. Stability Considerations in IV Drug Preparation and Use, in Manual of Home Parenteral Therapy, J. Neilson and G. Neilson, eds. 8 (2003).
- Prankerd, R.J. Aspartame, in Analytical Profiles of Drug Substances and Excipients, ed., H.G. Brittain (vol. 29, Academic Press, San Diego (2002) pp. 7-56).
- Preechagoon, D., Smith, M.T.S.and RJ Prankerd. Investigation of the antinociceptive efficacy and relative potency of long-acting injectable 3-acylmorphine-6-sulfate prodrugs in rats. Int J Pharm, 1998, 163, 191.
- Preechagoon, D., Brereton, I., Staatz, C. and Prankerd, R.J. 3-Acyl ester prodrugs of morphine-6-sulphate, a potent analgesic: syntheses, NMR spectra and some physico-chemical properties. Int J Pharm, 1998, 163, 177.
- Prankerd, R.J. and Elsabee, M. Thermal analysis of chiral drugs. The DSC behaviour of mixtures of ephedrine HCl and pseudoephedrine HCl enantiomers. Thermochimica Acta, 1995, 248, 147.
- Elsabee, M. and Prankerd, R.J. Solid state properties of drugs. Part III. Differential scanning calorimetry of drugs existing as racemic solid solutions, racemic mixtures and racemic compounds. Int J Pharm, 1992, 86, 221.
- Prankerd, R.J., Stone, H.W., Sloan, K.B. and Perrin, J.H. Degradation of aspartame in acidic aqueous media and its stabilization by complexation with cyclodextrin or modified cyclodextrins. Int J Pharm, 1992, 88, 189.
- Prankerd, R.J. Solid state properties of drugs. Part I. Estimation of heat capacities for fusion and thermodynamic functions for solution from aqueous solubility-temperature dependence measurements. Int J Pharm, 1992, 84, 233.
- Prankerd, R.J. and McKeown, R.H. Physico-chemical properties of barbituric acid derivatives. Part I. Solubility-temperature dependence for 5,5-disubstituted barbituric acids in aqueous solutions. Int J Pharm, 1990, 62, 37.
- McKeown, R.H. and Prankerd, R.J. First thermodynamic dissociation constants of barbituric acids in water at 25°C. Part 3. 5,5-Alkylenebarbituric acids. A comparison with 5,5-dialkylbarbituric acids, and with mono- and di-carboxylic acids. J Chem Soc, (Perkin II), 1981, 481.
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